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Updated: Jul 9, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Negative and positive allosteric modulators of the P2X(7) receptor

A D Michel1, L J Chambers, D S Walter

  • 1Neurology Centre of Excellence for Drug Discovery, GlaxoSmithKline Research & Development Limited, Harlow, Essex, UK. anton.d.michel@gsk.com

British Journal of Pharmacology
|December 12, 2007
PubMed
Abstract

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