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Published on: June 8, 2017
Pharmacokinetics of dihydroartemisinin in a murine malaria model
Kevin T Batty1, Peter L Gibbons, Timothy M E Davis
1School of Pharmacy, Curtin University of Technology, Bentley, Western Australia. kevin.batty@curtin.edu.au
The American Journal of Tropical Medicine and Hygiene
|April 4, 2008
Abstract:
Pharmacokinetic properties of dihydroartemisinin (DHA) were determined in mice given 100 mg/kg intraperitoneal DHA. Half-life, CL/F, and V/F were 25 min, 61.3 L/hr/kg, and 36.3 L/kg in malaria-infected mice and 19 min, 50.9 L/hr/kg, and 23.0 L/kg in controls. These data are valuable for pharmacokinetic-pharmacodynamic evaluations of DHA in murine models.

