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Updated: Jul 5, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
10:33

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

An isoform-selective, small-molecule inhibitor targets the autoregulatory mechanism of p21-activated kinase

Sean W Deacon1, Alexander Beeser, Jami A Fukui

  • 1Basic Sciences Division, Fox Chase Cancer Center, Philadelphia, PA 19111, USA.

Chemistry & Biology
|April 19, 2008
PubMed

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