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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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1-[(Imidazolidin-2-yl)imino]indazole. Highly alpha 2/I1 selective agonist: synthesis, X-ray structure, and biological

Franciszek Saczewski1, Anita Kornicka, Apolonia Rybczyńska

  • 1Department of Chemical Technology of Drugs and Department of Pathophysiology, Medical University of Gdańsk, 80-416 Gdańsk, Poland. saczew@amg.gda.pl

Journal of Medicinal Chemistry
|June 4, 2008
PubMed

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