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Updated: Jul 4, 2026

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
10:33

Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

Published on: October 26, 2015

Locking the two ends of tetrapeptidic HTLV-I protease inhibitors inside the enzyme

Meihui Zhang1, Jeffrey-Tri Nguyen, Henri-Obadja Kumada

  • 1Department of Medicinal Chemistry, Center for Frontier Research in Medicinal Science and 21st Century COE Program, Kyoto Pharmaceutical University, Yamashina-ku, Kyoto 607-8412, Japan.

Bioorganic & Medicinal Chemistry
|June 19, 2008
PubMed

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