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Quantitative Structure-Activity Relationship, Activity Prediction, and Molecular Dynamics of Non-nucleotide Reverse Transcriptase Inhibitors
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Solution kinetics measurements suggest HIV-1 protease has two binding sites for darunavir and amprenavir

Andrey Y Kovalevsky1, Arun K Ghosh, Irene T Weber

  • 1Departments of Biology and Chemistry, Molecular Basis of Disease Program, Georgia State University, Atlanta, Georgia 30303, USA.

Journal of Medicinal Chemistry
|September 24, 2008
PubMed

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