[5-Acyloxydioxolanones as prodrugs of non-steroidal anti-inflammatory agents. 1]

¹Pharmazeutich-Chemisches Institut, Universität Heidelberg.

|May 1, 1991

Abstract:

The derivatissation of various acidic non-steroidal anti-inflammatory drugs to 5-acyloxy-1,3-dioxolan-4-ones is described. The synthesis of the title compounds is achieved by reaction of 5-bromo-1,3-dioxolan-4-ones with the salts of the carbonic acids.

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Abstract:

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