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Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides
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Design and synthesis of a beta-lactamase activated 5-fluorouracil prodrug

Ryan M Phelan1, Marc Ostermeier, Craig A Townsend

  • 1Department of Chemistry, Johns Hopkins University, 3400 N. Charles St., Baltimore, MD 21212, USA.

Bioorganic & Medicinal Chemistry Letters
|January 27, 2009
PubMed

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