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Second generation of BACE-1 inhibitors part 3: Towards non hydroxyethylamine transition state mimetics

Nicolas Charrier1, Brian Clarke, Leanne Cutler

  • 1Neurology and Gastrointestinal Centre of Excellence for Drug Discovery, GlaxoSmithKline R&D, New Frontiers Science Park, Third Avenue, Harlow, Essex CM19 5AW, United Kingdom.

Bioorganic & Medicinal Chemistry Letters
|May 2, 2009
PubMed

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