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Farnesyltransferase inhibitor as anticancer agent

Anuj G Agrawal1, Rakesh R Somani

  • 1Department of Pharmaceutical Chemistry, Bharati Vidyapeeth's College of Pharmacy, Sec-8, CBD, Navi Mumbai-400 614, India. royalanuj@rediffmail.com

Mini Reviews in Medicinal Chemistry
|June 13, 2009
PubMed
Summary

Targeting Ras farnesylation is crucial for cancer treatment, as inhibiting this process with farnesyltransferase inhibitors (FTIs) shows promise. FTIs, when combined with chemotherapy, can enhance anti-cancer effects.

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