cANF causes endothelial cell hyperpolarization by activation of chloride channels

Aaron Simon1, Gong Xin Liu, Gideon Koren

  • 1Vascular Research Laboratory, Providence VA Medical Center, Providence, RI 02908, USA.

Peptides
|August 18, 2009
PubMed
Abstract

Insights

Natriuretic peptide receptor-C (NPR-C) activation by cANF(4-23) causes endothelial cell hyperpolarization. This effect is mediated by chloride channels, independent of G(i) protein and PKG signaling pathways.

Area of Science:

  • Cardiovascular Physiology
  • Cellular Electrophysiology
  • Endothelial Cell Biology

Background:

  • Natriuretic peptides bind to NPR-C, influencing cellular function via G(i) protein complexes.
  • NPR-C activates K(+) and non-selective cation channels in vascular smooth muscle and cardiac fibroblasts.
  • The electrophysiological impact of NPR-C on endothelial cells (EC) remains unexamined.

Purpose of the Study:

  • To investigate the effect of cANF(4-23), a selective NPR-C ligand, on endothelial cell membrane potential (E(m)).

Main Methods:

  • Endothelial cell membrane potential changes were measured using non-invasive fluorescence imaging with DiBAC(4)(3).
  • Cells were exposed to cANF(4-23) with various ion channel and second messenger inhibitors.
  • NPR-C expression in rat lung microvascular endothelial cells was analyzed via RT-PCR.
  • Perforated patch clamp recordings were used to confirm ion current mechanisms.

Main Results:

  • cANF(4-23) induced significant endothelial cell hyperpolarization, indicated by decreased cellular fluorescence.
  • Hyperpolarization was not affected by inhibitors of K(+) channels, Ca(2+) channels, G(i) protein, or PKG.
  • Chloride (Cl(-)) channel inhibitors (4,4'-diisothiocyanatostilbene-2,2'-disulfonic acid, niflumic acid) and hypertonic saline attenuated the hyperpolarization.
  • Patch clamp confirmed a Cl(-) current mediated by cANF(4-23), inhibited by niflumic acid.
  • RT-PCR confirmed NPR-C expression in vascular smooth muscle cells but not in EC.

Conclusions:

  • cANF(4-23) induces endothelial cell hyperpolarization.
  • This hyperpolarization is primarily mediated by the activation of Cl(-) channels.
  • The mechanism is independent of G(i) protein and protein kinase G (PKG) signaling.

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