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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Dipeptide-derived nitriles containing additional electrophilic sites: potentially irreversible inhibitors of cysteine

Reik Löser1, Michael Gütschow

  • 1Pharmazeutisches Institut, Pharmazeutische Chemie I, Rheinische Friedrich-Wilhelms-Universität, Bonn, Germany. reikloeser@gmx.de

Journal of Enzyme Inhibition and Medicinal Chemistry
|November 17, 2009
PubMed

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