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Chemical Inactivation of the E3 Ubiquitin Ligase Cereblon by Pomalidomide-based Homo-PROTACs
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Chemical Inactivation of the E3 Ubiquitin Ligase Cereblon by Pomalidomide-based Homo-PROTACs

Published on: May 15, 2019

New thalidomide analogues derived through Sonogashira or Suzuki reactions and their TNF expression inhibition

Scott G Stewart1, Carlos J Braun, Sze-Ling Ng

  • 1The School of Biomedical, Biomolecular and Chemical Sciences, The University of Western Australia Crawley, WA 6009, Australia. sgs@cyllene.uwa.edu.au

Bioorganic & Medicinal Chemistry
|December 26, 2009
PubMed

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