Design, synthesis, and biological evaluation of novel estradiol-bisphosphonate conjugates as bone-specific estrogens

Masahiko Morioka1, Akihito Kamizono, Hirosato Takikawa

  • 1Medicinal Chemistry Laboratory, Research Division, Mitsubishi-Tanabe Pharma Corporation, 1000 Kamoshida-cho, Aoba-ku, Yokohama 227-0033, Japan.