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Updated: Jun 16, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission

Published on: August 16, 2018

Rapid P1 SAR of brain penetrant tertiary carbinamine derived BACE inhibitors

Hong Zhu1, Mary B Young, Philippe G Nantermet

  • 1Department of Medicinal Chemistry, Merck Research Laboratories, West Point, PA 19486, USA.

Bioorganic & Medicinal Chemistry Letters
|February 4, 2010
PubMed

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