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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK1 antagonists

Gregori J Morriello1, Sander G Mills, Tricia Johnson

  • 1Department of Medicinal Chemistry, Merck Research Laboratories, Rahway, NJ 07065, USA. greg_morriello@merck.com

Bioorganic & Medicinal Chemistry Letters
|February 16, 2010
PubMed

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