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The Development and Application of Biophysical Assays for Evaluating Ternary Complex Formation Induced by Proteolysis Targeting Chimeras (PROTACS)
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CHIPS binds to the phosphorylated N-terminus of the C5a-receptor

Anton Bunschoten1, Louris J Feitsma, John A W Kruijtzer

  • 1Medicinal Chemistry & Chemical Biology, Faculty of Science, Utrecht University, Sorbonnelaan 16, 3584 CA, Utrecht, The Netherlands.

Bioorganic & Medicinal Chemistry Letters
|May 12, 2010
PubMed

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