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Updated: Jun 12, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Strategy for the identification of GPR23/LPA4 receptor agonists and inverse agonists

Soo Hang Wong1, Rommel Mallari, Melissa Graham

  • 1Lead Discovery, Amgen Inc., Thousand Oaks, California 91320, USA.

Assay and Drug Development Technologies
|May 21, 2010
PubMed

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