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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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Design of 1-piperazinyl-4-arylphthalazines as potent Smoothened antagonists

Brian S Lucas1, Wade Aaron, Songzhu An

  • 1Department of Medicinal Chemistry, AMGEN, S. San Francisco, CA 94080, USA. blucas@amgen.com

Bioorganic & Medicinal Chemistry Letters
|May 25, 2010
PubMed

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