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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Small molecule antagonists of chemokine receptors--is promiscuity a virtue?

James E Pease1, Richard Horuk

  • 1Leukocyte Biology Section, National Heart and Lung Institute, Faculty of Medicine, Imperial College of Science, Technology & Medicine, South Kensington Campus, London SW7 2AZ, UK. j.pease@imperial.ac.uk

Current Topics in Medicinal Chemistry
|June 12, 2010
PubMed

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