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Real-Time Monitoring of Aurora kinase A Activation using Conformational FRET Biosensors in Live Cells
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Discovery of orally bioavailable imidazo[1,2-a]pyrazine-based Aurora kinase inhibitors

David B Belanger1, Michael J Williams, Patrick J Curran

  • 1Department of Medicinal Chemistry, Merck Research Laboratories, 320 Bent Street, Cambridge, MA 02141, USA. david.belanger@merck.com

Bioorganic & Medicinal Chemistry Letters
|September 22, 2010
PubMed

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