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Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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Novel structural insights for drug design of selective 5-HT(2C) inverse agonists from a ligand-biased receptor model

Nicolas Renault1, Arnaud Gohier, Philippe Chavatte

  • 1Faculté des Sciences Pharmaceutiques et Biologiques, Laboratoire de Chimie Thérapeutique, EA GRIIOT, Université Nord de France, 3 rue du Professeur Laguesse, BP 83, 59006 Lille Cedex, France.

European Journal of Medicinal Chemistry
|October 1, 2010
PubMed

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