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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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5-Piperazinyl-3-sulfonylindazoles as potent and selective 5-hydroxytryptamine-6 antagonists

Kevin G Liu1, Albert J Robichaud, Ronald C Bernotas

  • 1Wyeth Research, CN 8000, Princeton, New Jersey 08543, United States. liuk@lundbeck.com

Journal of Medicinal Chemistry
|October 12, 2010
PubMed

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