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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Magnesium coordination-directed n-selective stereospecific alkylation of 2-pyridones, carbamates, and amides using

Yuan-Qing Fang1, Matthew M Bio, Karl B Hansen

  • 1Department of Chemical Process Research & Development, Amgen Inc., 360 Binney Street, Cambridge, Massachusetts 02142, USA. yfang@amgen.com

Journal of the American Chemical Society
|October 21, 2010
PubMed

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