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Published on: February 20, 2018
Chemokine receptor CXCR3 promotes growth of glioma
Che Liu1, Defang Luo, Brent A Reynolds
1Department of Pharmacology and Therapeutics, College of Medicine, University of Florida, Gainesville, FL 32610, USA.
Abstract:
Human glioblastoma multiforme (GBM) is the most common primary brain tumor in adults. The poor prognosis and minimally successful treatments of GBM indicates a need to identify new therapeutic targets. In this study, we examined the role of CXCR3 in glioma progression using the GL261 murine model of malignant glioma. Intracranial GL261 tumors express CXCL9 and CXCL10 in vivo. Glioma-bearing CXCR3-deficient mice had significantly shorter median survival time and reduced numbers of tumor-infiltrated natural killer and natural killer T cells as compared with tumor-bearing wild-type (WT) mice. In contrast, pharmacological antagonism of CXCR3 with NBI-74330 prolonged median survival times of both tumor-bearing WT and CXCR3-deficient mice when compared with vehicle-treated groups. NBI-74330 treatment did not impact tumor infiltration of lymphocytes and microglia. A small percentage of GL261 cells were identified as CXCR3(+), which was similar to the expression of CXCR3 in several grade IV human glioma cell lines (A172, T98G, U87, U118 and U138). When cultured as gliomaspheres (GS), the human and murine lines increased CXCR3 expression; CXCR3 expression was also found in a primary human GBM-derived GS. Additionally, CXCR3 isoform A was expressed by all lines, whereas CXCR3-B was detected in T98G-, U118- and U138-GS cells. CXCL9 or CXCL10 induced in vitro glioma cell growth in GL261- and U87-GS as well as inhibited cell loss in U138-GS cells and this effect was antagonized by NBI-74330. The results suggest that CXCR3 antagonism exerts a direct anti-glioma effect and this receptor may be a potential therapeutic target for treating human GBM.
Insights
Targeting CXCR3 may offer a new therapeutic strategy for glioblastoma multiforme (GBM). Blocking CXCR3 with NBI-74330 prolonged survival in a mouse model, suggesting direct anti-glioma effects.
Area of Science:
- Neuroscience
- Immunology
- Oncology
Background:
- Glioblastoma multiforme (GBM) is an aggressive brain tumor with poor prognosis.
- Current treatments for GBM are minimally successful, highlighting the need for novel therapeutic targets.
Purpose of the Study:
- To investigate the role of C-X-C motif chemokine receptor 3 (CXCR3) in glioma progression.
- To evaluate CXCR3 antagonism as a potential therapeutic strategy for GBM.
Main Methods:
- Utilized the GL261 murine model of malignant glioma.
- Administered pharmacological CXCR3 antagonist NBI-74330 to tumor-bearing mice.
- Assessed cell growth and survival in vitro using human and murine glioma cell lines and gliomaspheres.
Main Results:
- Glioma-bearing CXCR3-deficient mice exhibited reduced survival and fewer tumor-infiltrated immune cells.
- Pharmacological antagonism of CXCR3 with NBI-74330 prolonged survival in both wild-type and CXCR3-deficient mice.
- CXCR3 antagonism demonstrated direct anti-glioma effects in vitro, including inhibition of glioma cell growth.
Conclusions:
- CXCR3 plays a significant role in glioma progression.
- CXCR3 antagonism represents a promising therapeutic target for human glioblastoma multiforme.
- Further research into CXCR3-targeted therapies for GBM is warranted.
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