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Updated: Jun 6, 2026

Methods for the Discovery of Novel Compounds Modulating a Gamma-Aminobutyric Acid Receptor Type A Neurotransmission
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4-aryl piperazine and piperidine amides as novel mGluR5 positive allosteric modulators

Hui Xiong1, Todd A Brugel, Michael Balestra

  • 1CNS Discovery, AstraZeneca Pharmaceuticals, Wilmington, DE, USA. hui.xiong@astrazeneca.com

Bioorganic & Medicinal Chemistry Letters
|November 12, 2010
PubMed

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