Design, synthesis, and structure-activity relationship study of bicyclic piperazine analogs of indole-3-carboxamides

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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles
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Preparation of Stable Bicyclic Aziridinium Ions and Their Ring-Opening for the Synthesis of Azaheterocycles

Published on: August 22, 2018

Elizabeth M Moir1, Kazuya Yoshiizumi, Jim Cairns

  • 1Department of Chemistry, Merck Research Laboratories, MSD Ltd, Newhouse, Lanarkshire, UK.

Bioorganic & Medicinal Chemistry Letters
|November 16, 2010
PubMed

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