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3-(Pyridin-2-yl-ethynyl)benzamide metabotropic glutamate receptor 5 negative allosteric modulators: hit to lead

Adam M Gilbert1, Matthew G Bursavich, Sabrina Lombardi

  • 1Pfizer Global Research and Development, Groton Laboratories, Eastern Point Road, Groton, CT 06340, USA. adam.gilbert@pfizer.com

Bioorganic & Medicinal Chemistry Letters
|December 4, 2010
PubMed

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