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Preparation of N-(2-alkoxyvinyl)sulfonamides from N-tosyl-1,2,3-triazoles and Subsequent Conversion to Substituted Phthalans and Phenethylamines
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N-(2,5-Dimethoxy-phen-yl)-4-nitro-benzene-sulfonamide

Guo-Yao Zhang1, Shan Qian, Xiao-Cen Li

  • 1Key Laboratory of Drug Targeting of the Education Ministry, West China School of Pharmacy, Sichuan University, Chengdu 610041, People's Republic of China.

Acta Crystallographica. Section E, Structure Reports Online
|May 18, 2011
PubMed
Summary

This study details a chemical intermediate crucial for synthesizing beta-3 adrenergic receptor agonists. Molecular analysis reveals specific structural features and intermolecular interactions in its crystalline form.

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