Chronic CaMKII inhibition blunts the cardiac contractile response to exercise training

Guri Kaurstad1, Marcia N Alves, Ole J Kemi

  • 1K.G. Jebsen Center of Exercise in Medicine, Norwegian University of Science and Technology (NTNU), Trondheim, Norway.

Insights

Chronic Ca(2+)/calmodulin-dependent protein kinase II (CaMKII) inhibition with KN-93 enhanced exercise capacity in mice. However, it impaired cardiac function and blunted exercise benefits on cardiomyocyte shortening, revealing complex effects.

Area of Science:

  • Cardiovascular Physiology
  • Exercise Science
  • Molecular Cardiology

Background:

  • Ca(2+)/calmodulin-dependent protein kinase II (CaMKII) is crucial for cardiac function.
  • Understanding CaMKII's role in exercise adaptation is vital for cardiac health and disease management.

Purpose of the Study:

  • To investigate the impact of chronic CaMKII inhibition on cardiorespiratory function and cardiac performance during exercise training in healthy mice.
  • To elucidate the specific effects of KN-93, a CaMKII inhibitor, on exercise capacity and cardiac remodeling.

Main Methods:

  • Randomized controlled trial in mice with four groups: sham sedentary, sham exercise, KN-93 sedentary, and KN-93 exercise.
  • Cardiorespiratory fitness assessed via ergospirometry.
  • Cardiac function evaluated using echocardiography and cardiomyocyte contractility assays.

Main Results:

  • CaMKII inhibition (KN-93) alone did not affect exercise capacity or fractional shortening.
  • Exercise training significantly increased maximal oxygen uptake in KN-93 treated mice compared to sham mice (22% vs 8%).
  • KN-93 impaired exercise-induced improvements in in vivo fractional shortening and blunted cardiomyocyte fractional shortening response to training.

Conclusions:

  • Chronic CaMKII inhibition paradoxically enhances maximal oxygen uptake during exercise training.
  • CaMKII inhibition negatively impacts cardiac function and cardiomyocyte contractility, despite exercise.
  • The effects of CaMKII inhibition on cardiac function and exercise adaptation are complex and multifaceted.

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