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A Syngeneic Mouse Model of Metastatic Renal Cell Carcinoma for Quantitative and Longitudinal Assessment of Preclinical Therapies
Published on: April 12, 2017
Safety and efficacy of molecularly targeted agents in patients with metastatic kidney cancer with renal dysfunction
Sachin Gupta1, Venkata Parsa, Lance K Heilbrun
1Division of Hematology/Oncology, Karmanos Cancer Institute/Wayne State University, Detroit, Michigan 48201, USA.
Abstract:
Multiple molecularly targeted agents (MTAs) have been approved for the management of metastatic renal cell carcinoma (mRCC). Sunitinib and mammalian target of rapamycin inhibitors (temsirolimus, everolimus) are primarily metabolized in the liver, whereas the metabolism of bevacizumab is unclear. There are limited data on the toxicity profile and the efficacy of these agents in patients with renal insufficiency (RI). This is clinically relevant, especially as about one-third of patients with mRCC have renal dysfunction. The primary objective was to assess the safety and efficacy of targeted agents in patients with mRCC with RI. Medical records of patients with mRCC at Wayne State University, started on sunitinib, temsirolimus, everolimus, or bevacizumab, were reviewed. Patients with a calculated creatinine clearance of less than or equal to 60 ml/min were deemed to have RI. Data on safety and efficacy of MTA therapy were collected and analyzed with respect to renal function. RI was observed in 33% of our patients with mRCC. The incidence of toxicities, responses, time to progression, and overall survival were not significantly different in patients with RI compared with patients with normal renal function. Patients with RI had larger median increases in blood pressure with sunitinib and bevacizumab, increased incidence of thyroid dysfunction with sunitinib, and increased incidence of rash and dose interruptions with mammalian target of rapamycin inhibitors, than did patients with normal renal function. In conclusion, RI was commonly observed in our patients with mRCC. Molecularly targeted agents are well tolerated, and efficacy seems to be maintained in patients with RI. Vigilant monitoring of hypertension would be recommended for patients receiving sunitinib and bevacizumab.
Insights
Molecularly targeted agents (MTAs) are effective for metastatic renal cell carcinoma (mRCC) patients with renal insufficiency (RI). These treatments show similar efficacy and safety profiles, with careful blood pressure monitoring recommended for specific agents.
Area of Science:
- Oncology
- Nephrology
- Pharmacology
Background:
- Metastatic renal cell carcinoma (mRCC) management increasingly involves molecularly targeted agents (MTAs).
- Renal insufficiency (RI) affects approximately one-third of mRCC patients, yet data on MTA safety and efficacy in this population are limited.
- Key MTAs like sunitinib and mTOR inhibitors undergo hepatic metabolism, while bevacizumab metabolism is less understood.
Purpose of the Study:
- To evaluate the safety and efficacy of MTAs in mRCC patients with varying degrees of renal function.
- To identify any specific toxicities or efficacy differences associated with RI during MTA therapy.
Main Methods:
- Retrospective review of mRCC patients treated with sunitinib, temsirolimus, everolimus, or bevacizumab at Wayne State University.
- Patients were categorized based on creatinine clearance (≤60 ml/min for RI).
- Safety data (toxicities, dose interruptions) and efficacy outcomes (response rates, time to progression, overall survival) were analyzed concerning renal function.
Main Results:
- RI was present in 33% of the studied mRCC patient cohort.
- No significant differences in overall toxicity incidence, response rates, time to progression, or overall survival were observed between patients with RI and those with normal renal function.
- Patients with RI experienced greater increases in blood pressure with sunitinib and bevacizumab, and a higher incidence of thyroid dysfunction with sunitinib and rash/dose interruptions with mTOR inhibitors.
Conclusions:
- RI is a common comorbidity in mRCC patients.
- MTAs demonstrate maintained efficacy and are generally well-tolerated in patients with RI.
- Close monitoring for hypertension is advised for patients on sunitinib and bevacizumab, especially those with RI.
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