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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones
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A Direct, Regioselective and Atom-Economical Synthesis of 3-Aroyl-N-hydroxy-5-nitroindoles by Cycloaddition of 4-Nitronitrosobenzene with Alkynones

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Optimization of (arylpiperazinylbutyl)oxindoles exhibiting selective 5-HT₇ receptor antagonist activity

Balázs Volk1, István Gacsályi, Katalin Pallagi

  • 1Chemical Research Division, EGIS Pharmaceuticals Plc., P.O. Box 100, Budapest, H-1475 Hungary. volk.balazs@egis.hu

Journal of Medicinal Chemistry
|August 24, 2011
PubMed

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