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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors

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X-ray structures of checkpoint kinase 2 in complex with inhibitors that target its gatekeeper-dependent hydrophobic

George T Lountos1, Andrew G Jobson, Joseph E Tropea

  • 1Basic Science Program, SAIC-Frederick, Frederick, MD 21702-1201, USA.

FEBS Letters
|September 13, 2011
PubMed

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