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Substituted indole-1-acetic acids as potent and selective CRTh2 antagonists-discovery of AZD1981

Tim Luker1, Roger Bonnert, Steve Brough

  • 1Medicinal Chemistry, AstraZeneca R&D Charnwood, Loughborough, Leicestershire LE11 5RH, UK. tim.luker@astrazeneca.com

Bioorganic & Medicinal Chemistry Letters
|September 28, 2011
PubMed

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