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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
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Privileged scaffolds or promiscuous binders: a comparative study on rhodanines and related heterocycles in medicinal

Thomas Mendgen1, Christian Steuer, Christian D Klein

  • 1Medicinal Chemistry, Institute of Pharmacy and Molecular Biotechnology IPMB, Heidelberg University, Im Neuenheimer Feld 364, D-69120 Heidelberg, Germany.

Journal of Medicinal Chemistry
|November 15, 2011
PubMed

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