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Efficient Construction of Drug-like Bispirocyclic Scaffolds Via Organocatalytic Cycloadditions of α-Imino γ-Lactones and Alkylidene Pyrazolones
Published on: February 7, 2019
Francesco Giacalone1, Michelangelo Gruttadauria, Paola Agrigento
1Dipartimento di Scienze e Tecnologie Molecolari e Biomolecolari (STEMBIO) Sez. Chimica Organica E. Paternò, Università di Palermo, Viale delle Scienze, Ed. 17, 90128, Palermo, Italy.
Chiral organocatalysts are revolutionizing asymmetric synthesis with high activity and stereoselectivity. This review highlights advances in low-loading organocatalysts across diverse catalytic fields.
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