A trans diacyloxylation of indoles
Qiang Liu1, Qing Yong Zhao, Jie Liu
1College of Chemistry and Molecular Sciences, Wuhan University, Wuhan, 430072, PR China.
Abstract:
A trans diacyloxylation of indoles is accomplished by employing PhI(OAc)(2) as the oxidant. A broad range of functional groups are well tolerated. Both the electronic properties of the N-protecting groups of indoles and the acidity of the reaction media play important roles in the selectivity of indole acyloxylation reactions.
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