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Preparation of Enantiopure Non-Activated Aziridines and Synthesis of Biemamide B, D, and epiallo-Isomuscarine
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3-Phenyl-5-isothiazole carboxamides with potent mGluR1 antagonist activity

Matthew J Fisher1, Ryan T Backer, Vanessa N Barth

  • 1Lilly Research Laboratories, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, IN 46258, USA. fisher_matthew_j@lilly.com

Bioorganic & Medicinal Chemistry Letters
|March 6, 2012
PubMed

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