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Solid-phase Synthesis of [4.4] Spirocyclic Oximes
Published on: February 6, 2019
Solid-phase parallel synthesis of drug-like artificial 2H-benzopyran libraries
1Research Institute of Pharmaceutical Sciences, College of Pharmacy, Kyungpook National University, Buk-gu, Daegu, Korea. tlee@knu.ac.kr
Molecules (Basel, Switzerland)
|May 11, 2012
Abstract:
This review covers the construction of drug-like 2H-benzopyrans and related libraries using solid-phase parallel synthesis. In this context, the preparation of substituted benzopyrans such as mono-, di- and trisubstituted benzopyran derivatives and additional ring-fused benzopyrans such as benzopyranoisoxazoles, benzopyranopyrazoles, six-membered ring-fused benzopyrans, and polycyclic benzopyrans are highlighted.
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