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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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Functional and binding kinetic studies make a distinction between OX1 and OX2 orexin receptor antagonists

Stefania Faedo1, Elisabetta Perdonà, Marinella Antolini

  • 1Neurosciences Centre of Excellence for Drug Discovery, GlaxoSmithKline, Medicines Research Centre, 37135 Verona, Italy.

European Journal of Pharmacology
|July 17, 2012
PubMed

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