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Updated: May 18, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
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A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

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Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors

Stefanie Thiele1, Mikkel Malmgaard-Clausen, Jens Engel-Andreasen

  • 1Department of Neuroscience and Pharmacology, Faculty of Health and Medical Sciences, The Panum Institute, University of Copenhagen, Blegdamsvej 3, Dk-2200 Copenhagen, Denmark.

Journal of Medicinal Chemistry
|September 11, 2012
PubMed

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