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Optimization of an ether series of mGlu5 positive allosteric modulators: molecular determinants of MPEP-site

Jason T Manka1, Paige N Vinson, Karen J Gregory

  • 1Department of Pharmacology, Vanderbilt University Medical Center, Nashville, TN 37232, USA.

Bioorganic & Medicinal Chemistry Letters
|September 18, 2012
PubMed

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Cooperative Allosteric Transitions01:58

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Cooperative Allosteric Transitions01:58

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