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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Substrate-selective inhibition of protein kinase PDK1 by small compounds that bind to the PIF-pocket allosteric

Katrien Busschots1, Laura A Lopez-Garcia, Carmen Lammi

  • 1Research Group PhosphoSites, Department of Internal Medicine I, Universitätsklinikum Frankfurt, Theodor-Stern-Kai 7, 60590 Frankfurt, Germany.

Chemistry & Biology
|September 25, 2012
PubMed

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