Emerging roles of Nrf2 and phase II antioxidant enzymes in neuroprotection

Meijuan Zhang1, Chengrui An, Yanqin Gao

  • 1State Key Laboratory of Medical Neurobiology and Institute of Brain Science, Fudan University, Shanghai, China.

Progress in Neurobiology
|October 3, 2012
PubMed

Insights

Phase II enzymes detoxify harmful substances and are regulated by the Keap1/Nrf2 pathway. Their altered expression in neurological diseases suggests potential as therapeutic targets for neuroprotection.

Area of Science:

  • Biochemistry
  • Neuroscience
  • Toxicology

Background:

  • Phase II metabolic enzymes detoxify xenobiotics, increasing hydrophilicity for excretion.
  • These enzymes are crucial in preventing mutagen and carcinogen damage.
  • The Keap1/Nrf2/ARE pathway regulates phase II enzyme expression.

Purpose of the Study:

  • To review the role of phase II genes in the central nervous system (CNS).
  • To explore the neuroprotective effects of phase II enzymes.
  • To discuss the therapeutic potential of Nrf2 inducers for neurological diseases.

Main Methods:

  • Literature review focusing on phase II enzymes and the CNS.
  • Discussion of phase II enzyme expression, regulation, inducers, and executors.
  • Analysis of studies on neuroprotection conferred by phase II gene overexpression.

Main Results:

  • Altered expression of phase II genes is observed in postmortem CNS tissue of neurological disease patients.
  • Overexpression of phase II genes demonstrates neuroprotective effects in vitro and in vivo.
  • The Nrf2 pathway is a key regulator of these protective mechanisms.

Conclusions:

  • Phase II enzymes play a significant role in the CNS and in the pathogenesis of neurological disorders.
  • Targeting phase II genes, particularly via Nrf2 inducers, offers a promising therapeutic strategy for neurological diseases.
  • Further research is warranted to fully elucidate and leverage the neuroprotective potential of phase II enzymes.

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