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Development of Inhibitors of Protein-protein Interactions through REPLACE: Application to the Design and Development Non-ATP Competitive CDK Inhibitors
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Isatin replacements applied to the highly selective, muscarinic M1 PAM ML137: continued optimization of an MLPCN

Bruce J Melancon1, Michael S Poslusney, Patrick R Gentry

  • 1Department of Pharmacology, Vanderbilt University Medical Center, Nashville, TN 37232, USA.

Bioorganic & Medicinal Chemistry Letters
|December 15, 2012
PubMed

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