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Naphthyridinone (NTD) integrase inhibitors: N1 protio and methyl combination substituent effects with C3 amide groups

Brian A Johns1, Takashi Kawasuji, Jason G Weatherhead

  • 1GlaxoSmithKline Research & Development, Infectious Diseases Therapy Area Unit, Five Moore Drive, Research Triangle Park, NC 27709, USA. brian.a.johns@gsk.com

Bioorganic & Medicinal Chemistry Letters
|December 19, 2012
PubMed

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