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Updated: May 14, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Structure-based discovery of cellular-active allosteric inhibitors of FAK

Naoki Tomita1, Yoko Hayashi, Shinkichi Suzuki

  • 1Pharmaceutical Research Division, Takeda Pharmaceutical Company Ltd, 26-1 Muraoka-Higashi 2-Chome, Fujisawa, Kanagawa 251-8555, Japan. naoki.tomita@takeda.com

Bioorganic & Medicinal Chemistry Letters
|February 19, 2013
PubMed

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