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Updated: May 13, 2026

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators
07:41

A Kinetic Fluorescence-based Ca2+ Mobilization Assay to Identify G Protein-coupled Receptor Agonists, Antagonists, and Allosteric Modulators

Published on: February 20, 2018

Discovery of allosteric modulators of factor XIa by targeting hydrophobic domains adjacent to its heparin-binding

Rajesh Karuturi1, Rami A Al-Horani, Shrenik C Mehta

  • 1Department of Medicinal Chemistry and Institute for Structural Biology and Drug Discovery, Virginia Commonwealth University, Richmond, Virginia 23298, USA.

Journal of Medicinal Chemistry
|March 5, 2013
PubMed

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