Selective CB2 agonists with anti-pruritic activity: discovery of potent and orally available bicyclic 2-pyridones

Ken-ichi Kusakabe1, Yasuyoshi Iso, Yukio Tada

  • 1Medicinal Research Laboratories, Shionogi Pharmaceutical Research Center, 11-1 Futaba-cho 3-chome, Toyonaka, Osaka 561-0825, Japan. ken-ichi.kusakabe@shionogi.co.jp

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