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Regioselective O-Glycosylation of Nucleosides via the Temporary 2',3'-Diol Protection by a Boronic Ester for the Synthesis of Disaccharide Nucleosides
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C-Glucosides with heteroaryl thiophene as novel sodium-dependent glucose cotransporter 2 inhibitors

Yuichi Koga1, Shigeki Sakamaki, Mitsuya Hongu

  • 1Medicinal Chemistry Research Laboratories, Mitsubishi Tanabe Pharma Corporation, 2-2-50 Kawagishi, Toda, Saitama 335-8505, Japan.

Bioorganic & Medicinal Chemistry
|July 2, 2013
PubMed

Keywords:
CanagliflozinGlucosideSGLT2 inhibitorThiopheneType 2 diabetes

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